Chang Y, Zhang X, Horton JR, Spannhoff A, Bedford MT, Cheng S. Structural basis for inhibition of G9a and GLP histone lysine methyltransferases by BIX-01294. Nat Struct Mol Biol. e-Pub 2/2009.

Mai A, Cheng D, Bedford MT, Valente S, Nebbioso A, Perrone A, Brosch G, Sbardella G, De Bellis F, Miceli M, Altucci L. Epigenetic multiple ligands: Mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors. J Med Chem 51:2279-2290, 2008.

Mai A, Valente S, Cheng D, Perrone A, Ragno R, Simeoni S, Sbardella G, Brosch G, Nebbioso A, Conte M, Altucci L, and Bedford MT. Synthesis and biological validation of novel synthetic histone/protein methyltransferase inhibitors. Chem Med Chem 2:987-991, 2007.

Cheng D, Yadav N, King RW, Swanson MS, Weinstein EJ, Bedford MT. Small molecule regulators of protein arginine methyltransferases. J Biol Chem 279:23892-23899, 2004.